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Isku-darka 7P budada (1890208-58-8)

Budada 'Raw Compound 7P' oo kor u qaadeysa duruufaha neurite ee neurons aasaasiga ah ee aasaasiga ah oo laga soo qaatay hippocampus, kilkral cerebral, iyo retina. Qaabka xayawaanka ee dhaawaca dareemayaasha indhaha, Raw Compound 7P budada ayaa la muujiyey inay kadhigto koritaanka farqiga-43 axons oo togan, taasoo muujineysa in firfircoonida firfircoonida ee fitnada neerite ee Raw Compound 7P budada ay u tarjumeyso kicinta dib-u-cusboonaysiinta axon ee vivo.

Soo-saar: Soosaaris Dufcaddii
Xidhmada: 1KG / bac, 25KG / durbaan
Caqligu wuxuu awood u leeyahay inuu soo saaro oo uu bixiyo tiro badan. Dhammaan wax soo saarka ee hoos yimaada xaaladda cGMP iyo nidaamka xakamaynta tayada adag, dhammaan dukumeentiyada imtixaanka iyo muunada la heli karo.

Isku-darka budada 7P (1890208-58-8) fiidiyow

 

Isku-darka 7P budada Macluumaadka Saldhigga

magaca Isugeynta budada 7P
CAS 1890208-58-8
xagiisayna 98%
Magaca kiimikada 2-[(2-methoxyphenyl)[(4-methylphenyl)sulfonyl]amino]-N-(4-methoxy-3-pyridinyl)acetamide
Isku mid ahaanshaha Isdhaafka 7P

CHEMBL3824120

Formula kelli C22H23N3O5S
Miisaanka kelli 441.5 g / mol
Dhibicda Biyaha Qiyaastii 159 ℃
Muhiimadda InChI NAXWKPFXCOBXLE-UHFFFAOYSA-N
Form Solid
Imaanshaha White
Nolosha badh 1-2h
milmi Dhibaato ku jirta ethyl acetate, dichloromethan;

Si tartiib tartiib ah ayey ugu milmaysan tahay methanol;

biyaha

kaydinta Xaaladda Meel qalalan, oo iftiinka ka bax.
Codsiga Compound 7p waxaa loo soo saaray sidii mid ka mid ah taxaneyaal xeryo ah iyada oo ujeedadu tahay in la garto labada-hawlgale ee thromboxane receptor antagonist / synthase inhibitors.
Dukumentiga Tijaabinta Available

 

Isku-darka 7P budada Tilmaanta Guud

Budada 'Raw Compound 7P' oo kor u qaadeysa duruufaha neurite ee neurons aasaasiga ah ee aasaasiga ah oo laga soo qaatay hippocampus, kilkral cerebral, iyo retina.

Moodh xayawaan ah oo ku saabsan dhaawaca dareemayaasha indhaha, Raw Compound 7P waxaa lagu muujiyey inuu kicinayo koritaanka farqiga-43 axons togan, taasoo muujineysa in firfircoonida firfircoonida ee fitnada neerite ee Raw Compound 7P ay u tarjumeyso dhiirrigelinta dib-u-cusboonaysiinta axon ee vivo.

 

Isugeynta 7P (1890208-58-8) Taariikh

Compound 7p waxaa loo soo saaray sidii mid ka mid ah taxaneyaal xeryo ah iyada oo ujeedadu tahay in la garto labada-hawlgale ee thromboxane receptor antagonist / synthase inhibitors.

Xaqiiqdii xarunta 7p waxay muujineysaa xulashada prostaglandin I2 synthase (PTGIS, CYP8A1) oo ka sarreysa thromboxane synthase (CYP5A1).

 

Isku-darka 7P (1890208-58-8) Faa'iidooyinka

  1. Isbarbar dhig dareenka madaxa qoob ka ciyaarka
  2. Waxay kor u qaadaa dusha sare ee neurronimada neerfayaasha aasaasiga ah ee asaasiga ah oo laga soo qaatay hippocampus, cortex cerebral, iyo retina.

 

Isku-darka 7P (1890208-58-8) Daraasad dheeri ah

U habeyn dheeraad ah ee xarunta 7p iyo ballaarinta farsamooyinka ay ku adeegsato dib-u-cusboonaysiinta qalliinka ee vivo waxay bixin doontaa saldhig macquul ah dadaallada mustaqbalka lagu xoojinayo istiraatiijiyadaha daaweynta.

 

Isugeynta 7P (1890208-58-8) Tixraac

  • Naqshadeynta, isku-darka iyo isku-darka molikula ee thiazolidinedione waxay ku saleysantahay aasaaska benzene sulphonamide oo ay kujirto maadada loo yaqaan 'pyrazole core' sida wakiilada ka hortagga cudurka sonkorowga. Naim MJ, Alam O, Alam MJ, Hassan MQ, Siddiqui N, Naidu VGM, Alam MI. Kiimikada loo yaqaan 'Bioorg Chem'. 2018 Feb; 76: 98-112. doi: 10.1016 / j.bioorg.2017.11.010. Epub 2017 Nov 16. PMID: 29169079
  • Noocyada 1,3,5-triazine-ka soosaartay ayaa kudhaawacan kansarka kahortaga xubinta taranka dumarka ayagoo wax ka badalaya muujinta Bax, Bcl2 iyo Caspases. Wang X, Yi Y, Lv Q, Zhang J, Wu K, Wu W, Zhang W. Chem Biol Drug Des. 2018 Mar; 91 (3): 728-734. doi: 10.1111 / cbdd.13133. Epub 2017 Nov 15. PMID: 29068538
  • Waxyaabaha suurtagalka ah ee ka-hortagga kansarka ee 7-O-pentyl quercetin: Wax ku ool ah, xakamaynta-xuubka ka-hortagga xuub-ku-saleysan iyo saameyn-ku-sumowga. Sassi N, Mattarei A, Espina V, Liotta L, Zoratti M, Paradisi C, Biasutto L. Pharmacol Res. 2017 Okt; 124: 9-19. doi: 10.1016 / j.phrs.2017.07.016. Epub 2017 Jul 17. PMID: 28728925
  • Indole carboxylic acid esters oo ah melampomagnolide B waa wakiilada xinjirowga xinjirowga lidka ku ah labada unugyada dhiiga iyo burooyinka adag. Bommagani S, Ponder J, Penthala NR, Janganati V, Jordan CT, Borrelli MJ, Crooks PA. Eur J Med Chem. 2017 Og 18; 136: 393-405. doi: 10.1016 / j.ejmech.2017.05.031. Epub 2017 May 11. PMID: 28525840 Qodobka PMC ee Bilaashka ah
  • Tilmaamaha Kuufiyeyaasha ee ugu fiican ee loo yaqaan 'Nootropic Stack Guide': Wax kasta oo aad u Baahan Tahay Inaad Ogaato

 

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