Products

Budada HBT1 (489408-02-8)

Budada HBT1 waa AMPA-R [alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA) receptor] potentiator kaas oo kiciya soosaarka maskaxda maskaxda ka soo baxda (BDNF) wuxuuna muujiyaa saameyn yar oo agonistic ah neurons aasaasiga ah. HBT1 waxay ku xiraysaa aagga ligand-ku xiraya AMPA-R hab ku tiirsanaanta glutamate.

Soo-saar: Soosaaris Dufcaddii
Xidhmada: 1KG / bac, 25KG / durbaan
Caqligu wuxuu awood u leeyahay inuu soo saaro oo uu bixiyo tiro badan. Dhammaan wax soo saarka ee hoos yimaada xaaladda cGMP iyo nidaamka xakamaynta tayada adag, dhammaan dukumeentiyada imtixaanka iyo muunada la heli karo.

HBT1 Powder (489408-02-8) fiidiyaha

 

HBT1 Powder (489408-02-8) Saldhigga Macluumaadka

magaca Budada HBT1
CAS 489408-02-8
xagiisayna 98%
Magaca kiimikada 2-(((5-Methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl)acetyl)amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
Isku mid ahaanshaha HBT1; HBT-1; HBT 1
Formula kelli C16H17F3N4O2S
Miisaanka kelli 386.39
Dhibicda Biyaha /
Muhiimadda InChI PHLXSNIEQIKENK-UHFFFAOYSA-N
Form budo
Imaanshaha caddaan ah si beige ah
Nolosha badh /
milmi DMSO: 2 mg / mL, cad
kaydinta Xaaladda 0 - 4 C muddo gaaban (maalmo illaa toddobaadyo), ama -20 C muddo dheer (bilo).
Codsiga Awoodda soo dhoweynta AMPA
Dukumentiga Tijaabinta Available

 

HBT1 Powder (489408-02-8) Sifeynta Guud

Budada HBT1 waa awood qaata AMPA oo leh saameyn hoose oo agonistic ah, iyada oo laga fogaanayo jawaab celinta qaab-jalaatada ee wax-soo-saarka BDNF. Waa AMPA-R [alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA) reseptor] awood leh oo soo saarta wax soosaarka maskaxda ka soo baxda neurotrophic factor (BDNF) waxayna muujisaa saameyn yar oo agonistic ah neerfaha. HBT1 waxay kuxirantahay qaybta isku xidhka 'AMPA-R' ee habka ku tiirsanaanta glutamate.

 

HBT1 Powder (489408-02-8) Tixraac

[1] Kunugi A, Tajima Y, Kuno H, Sogabe S, Kimura H. HBT1, oo ah Novel AMPA Receptor Potentiator oo leh Saameynta Agonistic Hoose, Ka Fogaanshaha Jawaab-Baalan qaab-dhismeed ee Soosaarida Vitro BDNF. J Pharmacol Exp Ther. 2018 Mar; 364 (3): 377-389. doi: 10.1124 / jpet.117.245050. Epub 2018 Jan 3. La daabacay PMID: 29298820.
 

Maqaallada Daalacanaya